Pharmacology Weekly's: Comprehensive Drug Table of Substrates, Inhibitors, and Inducers of CYP450, UGT, and Transporters: A-B

Clinical Resources

Drugs: A-B, C-D, E-G, H-K, L-N, O-R, S-T, U-Z

COMPREHENSIVE DRUG REFERENCE TABLE: A-B ©2011 Pharmacology Weekly, Inc.
	CYP450 ENZYMES			UGT ENZYMES			TRANSPORTERS
DRUG	Substrate	Inhibitor	Inducer	Substrate	Inhibitor	Inducer	Substrate	Inhibitor	Inducer
5-FU		2C9					OAT2 BCRP MRP5
Abiraterone	3A4	2D6
Acetaminophen	1A2 2E1			1A1 1A6 1A9
Acetolol							P-gp
Acyclovir							OAT1 OCT1
Adefovir							OAT1 MRP1
Adriamycin							OCTN1
Alcohol
Aldosterone							P-gp
Alfentanil
Alfentanil	3A4
Alfuzosin	3A4
Aliskiren	3A4						P-gp
Allopurinol							OAT2
Almokalant				1A9 2B7
Almotriptan	3A4
Alosetron
Alprazolam	3A4
Alprenolol	2D6
Amantadine							OCT1 OCT2
Amiodarone	2C8 3A4	2B6 2C9 2D6 3A4					P-gp	P-gp
Amitriptyline	1A2 2C9 2D6 3A4			1A3 1A4				P-gp
Aminoglutethimide
Amlodipine	3A4
Amodiaquine	2C8
Amoxicillin							PEPT1 PEPT2
Ampicillin							PEPT1 PEPT2
Amprenavir	3A4	3A4	3A4				P-gp		P-gp
Amphetamine	2D6
Anagrelide
Anastrozole		2C8
Androsterone				1A4
Aprepitant	3A4	3A4	2C9
Aripiprazole	2D6 3A4
Ascorbic acid							OAT2
Artemisinin
Asenapine	1A2 2D6 3A4			1A4
Astemizole	3A4							P-gp
Atazanavir	3A4	1A2 2C9 3A4			1A1			BCRP
Atomoxetine	2D6
Atorvastatin	3A4			1A1 1A3 2B7			OATP1B1 BCRP P-gp	OATP1B1 BCRP P-gp
Azapropazone
Azithromycin
AZT							BCRP
Barbiturates		2B6 2C9 3A4	2B6 2C9 2C19 3A4			2B4 2B7 2B15
Bendamustine	3A4
Benzphetamine	2C8
Benzylpenicillin							OAT1
Bepridil	3A4
Bexarotene	3A4
Bifuralol	2D6
Bisoprolol	2D6
Boceprevir	3A4	3A4					P-gp	P-gp
Bromocriptine	3A4							P-gp
Budesonide	3A4
Bumetanide							OAT2
Buprenorphine	3A4
Bupropion	2B6	2D6
Buspirone	3A4

To view the individual tables for each of the CYP450 enzymes, UGT enzymes, or transporters click here